SCHEMBL3916689

SCHEMBL3916689

COc1ccc(C2(NS(C)(=O)=O)CNC(=O)N2CCCc2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.43
MMP1 P03956 4/20 0.42
MMP9 P14780 2/20 0.42
MMP13 P45452 2/20 0.42
ADAM17 P78536 2/20 0.42
KCNA5 P22460 3/20 0.41
KCNH2 Q12809 3/20 0.41
THRB P10828 1/20 0.41
OPRM1 P35372 1/20 0.41
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM3 P20309 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MMP2 P08253 2/20 0.38
MMP3 P08254 2/20 0.38
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3918962 0.95 KCNA5 (0.45) SIGMAR1MMP1MMP9MMP13ADAM17
SCHEMBL3917221 0.89 KCNA5 (0.45) SIGMAR1MMP1MMP9MMP13KCNA5
SCHEMBL3925223 0.88 KCNA5 (0.49) KCNA5KCNH2
SCHEMBL4104548 0.86 OPRM1 (0.37) SIGMAR1OPRM1POLBMAPTSMN1; SMN2
SCHEMBL3914439 0.86 CA12 (0.43) SIGMAR1MMP1MMP9MMP13ADAM17
SCHEMBL3925559 0.85 SIGMAR1 (0.40) SIGMAR1KCNA5KCNH2OPRM1POLB
SCHEMBL3925362 0.85 KCNA5 (0.52) SIGMAR1MMP1MMP9MMP13ADAM17
SCHEMBL3926338 0.85 KCNA5 (0.47) SIGMAR1MMP1MMP9MMP13ADAM17
SCHEMBL3916954 0.84 KCNA5 (0.48) MMP1MMP9MMP13ADAM17KCNA5
SCHEMBL3916079 0.83 KCNA5 (0.48) SIGMAR1MMP1MMP9MMP13ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035392-A1 IMIDAZOLE KV1. 5 POTASSIUM CHANNEL INHIBITORS Wyeth a Corporation of the State of Delaware (US) 2009-03-18 EP disclosed
WO-2007149874-A1 IMIDAZOLIDINONE KV1.5 POTASSIUM CHANNEL INHIBITORS WYETH (US) 2007-12-27 WO disclosed