SCHEMBL3928261

SCHEMBL3928261

CCOC(=O)CCCc1ccc([N+](=O)[O-])cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.50
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 3/20 0.49
TDP1 Q9NUW8 2/20 0.49
RAB9A P51151 3/20 0.47
NPC1 O15118 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
MAPK1 P28482 1/20 0.44
KMT2A Q03164 1/20 0.44
GLA P06280 1/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
CYP2C19 P33261 1/20 0.42
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PKM P14618 1/20 0.42
HASPIN Q8TF76 1/20 0.41
BCL9 O00512 1/20 0.41
CTNNB1 P35222 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12526399 0.87 CYP2C19 (0.50) MAPTKDM4EALDH1A1TDP1RAB9A
SCHEMBL4187236 0.84 MAPT (0.51) MAPTKDM4EALDH1A1RAB9ANPC1
SCHEMBL3936383 0.81 CYP1A2 (0.43) MAPTALDH1A1SMN1; SMN2KMT2ACYP2C19
SCHEMBL29966397 0.81 ADRA2A (0.48) MAPTALDH1A1SMN1; SMN2KMT2ACYP2C19
SCHEMBL12526403 0.81 ADRA2A (0.48) MAPTALDH1A1SMN1; SMN2KMT2ACYP2C19
SCHEMBL6745383 0.80 CYP2C19 (0.46) MAPTKDM4EALDH1A1RAB9ANPC1
SCHEMBL17028594 0.80 CYSLTR2 (0.45) KDM4EALDH1A1SMN1; SMN2KMT2AGLA
SCHEMBL7188600 0.80 MAPT (0.55) MAPTKDM4EALDH1A1TDP1MAPK1
SCHEMBL3135029 0.79 L3MBTL1 (0.55) MAPTKDM4EALDH1A1TDP1RAB9A
SCHEMBL13555429 0.79 MAPT (0.49) MAPTRAB9ANPC1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007418-A1 NOVEL BRONCHODILATING ISOQUINOLINE AMIDES RESPIRATORIUS AB (SE) 2009-01-15 WO disclosed
WO-2009007418-A1 NOVEL BRONCHODILATING ISOQUINOLINE AMIDES RESPIRATORIUS AB (SE) 2009-01-15 WO disclosed