SCHEMBL3934162

SCHEMBL3934162

NC(=S)N1CCN(C(=O)O)CC1COc1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.46
CHRNB2 P17787 2/20 0.46
CHRNA4 P43681 2/20 0.46
CHRNA1 P02708 1/20 0.46
CHRNB1 P11230 1/20 0.46
CHRNB4 P30926 1/20 0.46
CHRNA3 P32297 1/20 0.46
CHRNB3 Q05901 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL779253 0.86 CHRNA7 (0.44) CHRNA7CHRNB2CHRNA4CHRNA1CHRNB1
SCHEMBL3930902 0.85 NPSR1 (0.48) CHRNA7CHRNB2CHRNA4CHRNA1CHRNB1
SCHEMBL3937435 0.82 CHRNA1 (0.44) CHRNA7CHRNB2CHRNA4CHRNA1CHRNB1
SCHEMBL15841980 0.82 CHRNA7 (0.58) CHRNA7
SCHEMBL3939444 0.80 CHRNA7 (0.51) CHRNA7
SCHEMBL3931014 0.80 DRD2 (0.41) CHRNA7CHRNB2CHRNA4CHRNA1CHRNB1
SCHEMBL3930962 0.79 ALDH1A1 (0.43) CHRNA7CHRNB2CHRNA4CHRNA1CHRNB1
SCHEMBL4170987 0.79 ALDH1A1 (0.46) CHRNA7CHRNB2CHRNA4CHRNA1CHRNB1
SCHEMBL15841933 0.79 RECQL (0.47) CHRNA7CHRNB2CHRNA4CHRNA1CHRNB1
SCHEMBL4010198 0.79 CHRNA1 (0.41) CHRNA7CHRNB2CHRNA4CHRNA1CHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044038-A2 NOVEL PIPERAZINES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF Cornerstone Therapeutics Inc. (US) 2009-04-08 EP disclosed
WO-2007146066-A2 NOVEL PIPERAZINES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF CRITICAL THERAPEUTICS, INC. (US) 2007-12-21 WO disclosed