SCHEMBL3934451

SCHEMBL3934451

CC(=O)Nc1ncc(N)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
KDM4E B2RXH2 1/20 0.41
PTK2 Q05397 1/20 0.41
PGK1 P00558 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
PIK3CA P42336 2/20 0.39
GAA P10253 1/20 0.37
SCN9A Q15858 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
MTOR P42345 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11446331 0.82 PTK2 (0.51) ALDH1A1SMN1; SMN2KDM4EPTK2L3MBTL1
SCHEMBL9198708 0.79 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2KDM4EPTK2PGK1
SCHEMBL913171 0.79 L3MBTL1 (0.39) ALDH1A1SMN1; SMN2KDM4EPTK2CA1
SCHEMBL9648858 0.78 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2KDM4EPTK2L3MBTL1
SCHEMBL10388715 0.78 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2KDM4EPTK2PGK1
SCHEMBL3934366 0.77 CYP1A2 (0.40) ALDH1A1KDM4EL3MBTL1PIK3CATDP1
SCHEMBL9646715 0.77 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2KDM4EPTK2PGK1
SCHEMBL9646590 0.77 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2KDM4EPTK2PGK1
SCHEMBL3590963 0.76 GRM4 (0.41) ALDH1A1SMN1; SMN2KDM4EGAAMEN1
SCHEMBL28110473 0.76 ALDH1A1 (0.74) ALDH1A1SMN1; SMN2KDM4EL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831198-B1 PYRIDINE CARBOXAMIDE DERIVATIVES FOR USE AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2009-04-08 EP disclosed
CN-101128454-A Pyridine carboxamide derivatives for use as anticancer agents ASTRAZENECA AB (SE) 2008-02-20 CN disclosed