SCHEMBL3934495

SCHEMBL3934495

CN(C)CCNC(=O)c1ccc(Br)cc1F.O=C(O)c1ccc(Br)cc1F

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.65
SIGMAR1 Q99720 1/20 0.65
CYP1A2 P05177 1/20 0.61
ALDH1A1 P00352 6/20 0.53
KDM4E B2RXH2 3/20 0.53
HPGD P15428 3/20 0.53
ALOX12 P18054 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.51
HTT P42858 1/20 0.51
ACKR3 P25106 1/20 0.48
RAD52 P43351 1/20 0.45
PPARD Q03181 1/20 0.44
KMT2A Q03164 2/20 0.44
LMNA P02545 2/20 0.44
GAA P10253 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
DGAT1 O75907 1/20 0.43
HSD17B10 Q99714 2/20 0.42
GLA P06280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2926409 0.95 CYP1A2 (0.67) TMEM97SIGMAR1CYP1A2ALDH1A1KDM4E
SCHEMBL4077983 0.84 TMEM97 (0.58) TMEM97SIGMAR1CYP1A2ALDH1A1KDM4E
SCHEMBL26838419 0.82 TMEM97 (0.59) TMEM97SIGMAR1CYP1A2ALDH1A1KDM4E
SCHEMBL30231342 0.81 ACKR3 (0.69) TMEM97SIGMAR1CYP1A2ALDH1A1KDM4E
SCHEMBL2823242 0.80 CYP1A2 (0.68) TMEM97SIGMAR1CYP1A2ALDH1A1KDM4E
SCHEMBL12121026 0.80 HTT (0.74) TMEM97SIGMAR1CYP1A2ALDH1A1KDM4E
SCHEMBL582871 0.79 TMEM97 (0.57) TMEM97SIGMAR1CYP1A2ALDH1A1KDM4E
SCHEMBL18730432 0.79 SIGMAR1 (1.00) TMEM97SIGMAR1ACKR3
SCHEMBL17677968 0.79 CYP1A2 (0.49) TMEM97SIGMAR1CYP1A2ALDH1A1KDM4E
SCHEMBL2993559 0.79 HTT (0.56) TMEM97SIGMAR1CYP1A2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044058-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2009-04-08 EP disclosed
WO-2007148070-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2007-12-27 WO disclosed