SCHEMBL3938458

SCHEMBL3938458

C=CCCC(CC=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.37
GABBR2 O75899 2/20 0.33
GABBR1 Q9UBS5 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP2D6 P10635 2/20 0.33
CYP1A2 P05177 1/20 0.33
PKM P14618 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 2/20 0.31
HRH1 P35367 2/20 0.31
MAPK1 P28482 1/20 0.31
OPRD1 P41143 1/20 0.31
HTR2A P28223 1/20 0.31
RIPK1 Q13546 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL253606 0.83 CYP2C19 (0.52) CYP2C19SMN1; SMN2GABBR2GABBR1ALDH1A1
SCHEMBL3140559 0.80 CYP2D6 (0.42) CYP2C19SMN1; SMN2GABBR2GABBR1ALDH1A1
SCHEMBL23411628 0.78 ATM (0.39) CYP2C19GABBR2GABBR1ALDH1A1KDM4E
SCHEMBL9254662 0.78 TRPA1 (0.42) CYP2C19SMN1; SMN2GABBR2GABBR1ALDH1A1
SCHEMBL18642721 0.78 GABBR2 (0.47) CYP2C19SMN1; SMN2GABBR2GABBR1ALDH1A1
SCHEMBL2132327 0.78 LMNA (0.41) CYP2C19SMN1; SMN2ALDH1A1CYP2D6LMNA
SCHEMBL12654678 0.78 GABBR2 (0.35) CYP2C19SMN1; SMN2GABBR2GABBR1ALDH1A1
SCHEMBL1546516 0.78 AOC3 (0.40) CYP2C19SMN1; SMN2GABBR2GABBR1CYP2D6
SCHEMBL6802502 0.78 CYP2C19 (0.42) CYP2C19SMN1; SMN2GABBR2GABBR1ALDH1A1
SCHEMBL4908362 0.78 LMNA (0.41) CYP2C19SMN1; SMN2ALDH1A1CYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2043644-A1 NF- B INHIBITOR Otsuka Pharmaceutical Co., Ltd. (JP) 2009-04-08 EP disclosed
WO-2008010601-A1 NF- ϰB INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-01-24 WO disclosed