SCHEMBL3944112

SCHEMBL3944112

O=C(CC=Cc1c(F)cccc1F)CN1CCN(C2CCCCC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.47
KDM4E B2RXH2 6/20 0.47
ABCB1 P08183 1/20 0.45
RGS12 O14924 1/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TSHR P16473 2/20 0.42
MAPT P10636 2/20 0.42
HSD17B10 Q99714 2/20 0.42
ALOX12 P18054 1/20 0.42
TP53 P04637 1/20 0.42
ALOX15 P16050 1/20 0.42
MAPK1 P28482 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
MC4R P32245 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3944887 0.99 ALDH1A1 (0.45) ALDH1A1KDM4EABCB1RGS12MEN1
SCHEMBL3943715 0.86 ALDH1A1 (0.44) ALDH1A1KDM4EABCB1RGS12MEN1
SCHEMBL3945177 0.78 MAPT (0.49) ALDH1A1KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL3939893 0.77 ALDH1A1 (0.44) ALDH1A1KDM4ERGS12MEN1KMT2A
SCHEMBL3934180 0.77 TDP1 (0.38) ALDH1A1KDM4EKMT2ASMN1; SMN2HTT
SCHEMBL3935366 0.77 F2R (0.45) MEN1KMT2A
SCHEMBL1399126 0.74 ABCB1 (0.47) ALDH1A1KDM4EABCB1MEN1KMT2A
SCHEMBL1399128 0.74 ABCB1 (0.47) ALDH1A1KDM4EABCB1MEN1KMT2A
SCHEMBL1399145 0.73 ABCB1 (0.45) ALDH1A1KDM4EABCB1MEN1KMT2A
SCHEMBL1399143 0.73 ABCB1 (0.45) ALDH1A1KDM4EABCB1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2046748-A1 PHENYLPENTADIENOYL DERIVATIVES AND THEIR USE AS PAR 1 ANTAGONISTS Pierre Fabre Medicament (FR) 2009-04-15 EP claimed
WO-2007147822-A1 PHENYLPENTADIENOYL DERIVATIVES AND THEIR USE AS PAR 1 ANTAGONISTS PIERRE FABRE MEDICAMENT (FR) 2007-12-27 WO claimed