SCHEMBL3944601

SCHEMBL3944601

CN(CC(O)c1cccc(NC(=O)c2cccnc2)c1)C(=O)Oc1cnc(N(C)C)nc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.44
CSF1R P07333 4/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
ABL1 P00519 2/20 0.41
PDGFRB P09619 2/20 0.41
BCR P11274 2/20 0.41
SRC P12931 2/20 0.41
PDGFRA P16234 2/20 0.41
PRKCA P17252 2/20 0.41
PRKCD Q05655 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
PRKD3 O94806 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3944917 0.94 BACE1 (0.41) KCNK3CSF1RSMN1; SMN2HTTABL1
SCHEMBL3944650 0.89 KCNK3 (0.41) KCNK3CSF1RKMT2ANPC1RAB9A
SCHEMBL3951861 0.89 GRM4 (0.41) KCNK3SMN1; SMN2ABL1BCRSRC
SCHEMBL3946988 0.89 MEN1 (0.47) KCNK3SMN1; SMN2TSHRHTTPRKCD
SCHEMBL4154763 0.87 KCNK3 (0.41) KCNK3CSF1RKMT2A
SCHEMBL3952707 0.87 KCNK3 (0.41) KCNK3CSF1RTSHRKMT2ARAB9A
SCHEMBL3944465 0.85 KCNK3 (0.44) KCNK3SMN1; SMN2HTTABL1PDGFRB
SCHEMBL3951123 0.85 BACE1 (0.41) KMT2ANPC1RAB9AMEN1CYP1A2
SCHEMBL3951875 0.85 MAPT (0.42) KCNK3SMN1; SMN2HTTABL1PDGFRB
SCHEMBL3952248 0.84 BACE1 (0.40) PDGFRBSRCPDGFRAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed