SCHEMBL3952248

SCHEMBL3952248

CN(CC(O)c1cccc(NC(=O)NC(C)(C)C)c1)C(=O)Oc1cnc(N(C)C)nc1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.40
PDE4A P27815 1/20 0.36
AURKA O14965 1/20 0.34
RPS6KB1 P23443 1/20 0.34
FGFR1 P11362 3/20 0.33
SRC P12931 2/20 0.33
ALDH1A1 P00352 1/20 0.33
EGFR P00533 1/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
FGFR2 P21802 1/20 0.33
FGFR4 P22455 1/20 0.33
FGFR3 P22607 1/20 0.33
ALOX5 P09917 1/20 0.33
KDR P35968 1/20 0.33
BRAF P15056 1/20 0.33
CCR3 P51677 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3951123 0.90 BACE1 (0.41) BACE1AURKARPS6KB1ALOX5
SCHEMBL3944917 0.88 BACE1 (0.41) BACE1AURKARPS6KB1SRCPDGFRB
SCHEMBL3951861 0.86 GRM4 (0.41) BACE1SRCKDR
SCHEMBL3944465 0.84 KCNK3 (0.44) BACE1ALDH1A1EGFRPDGFRBPDGFRA
SCHEMBL3945805 0.84 LMNA (0.44) AURKARPS6KB1SRCALDH1A1PDGFRB
SCHEMBL3946482 0.84 ALOX5 (0.39) ALDH1A1ALOX5
SCHEMBL3944601 0.84 KCNK3 (0.44) SRCALDH1A1PDGFRBPDGFRA
SCHEMBL3944650 0.84 KCNK3 (0.41) BACE1ALDH1A1
SCHEMBL3951875 0.84 MAPT (0.42) BACE1SRCALDH1A1PDGFRBPDGFRA
SCHEMBL3946988 0.83 MEN1 (0.47) RPS6KB1FGFR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed