SCHEMBL4154763

SCHEMBL4154763

CN(CC(O)c1cccc(NC(=O)c2ccsc2)c1)C(=O)Oc1cnc(N(C)C)nc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.41
KCNK9 Q9NPC2 1/20 0.41
HPGD P15428 1/20 0.38
BACE1 P56817 1/20 0.38
AURKA O14965 1/20 0.35
RPS6KB1 P23443 1/20 0.35
TNIK Q9UKE5 1/20 0.34
ALOX5 P09917 1/20 0.33
GHSR Q92847 1/20 0.33
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GRM5 P41594 1/20 0.33
GNRHR P30968 1/20 0.33
MCHR1 Q99705 2/20 0.33
ATR Q13535 1/20 0.33
CSF1R P07333 1/20 0.33
KMT2A Q03164 2/20 0.33
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3944917 0.92 BACE1 (0.41) KCNK3KCNK9BACE1AURKARPS6KB1
SCHEMBL3951861 0.88 GRM4 (0.41) KCNK3KCNK9BACE1MAPT
SCHEMBL3944650 0.87 KCNK3 (0.41) KCNK3KCNK9BACE1MAPTGRM5
SCHEMBL3951875 0.87 MAPT (0.42) KCNK3KCNK9HPGDBACE1MAPT
SCHEMBL3944601 0.87 KCNK3 (0.44) KCNK3CSF1RKMT2A
SCHEMBL3946988 0.87 MEN1 (0.47) KCNK3KCNK9RPS6KB1MAPTKMT2A
SCHEMBL3952707 0.87 KCNK3 (0.41) KCNK3KCNK9BACE1AURKARPS6KB1
SCHEMBL3944465 0.85 KCNK3 (0.44) KCNK3KCNK9HPGDBACE1MAPT
SCHEMBL3951123 0.84 BACE1 (0.41) BACE1AURKARPS6KB1ALOX5KMT2A
SCHEMBL3952248 0.83 BACE1 (0.40) BACE1AURKARPS6KB1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed