SCHEMBL3944650

SCHEMBL3944650

CN(CC(O)c1cccc(NC(=O)c2cccc(Cl)c2)c1)C(=O)Oc1cnc(N(C)C)nc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 2/20 0.41
KCNK9 Q9NPC2 2/20 0.41
GRM5 P41594 2/20 0.40
CES1 P23141 1/20 0.39
MAPT P10636 3/20 0.39
TP53 P04637 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
BACE1 P56817 1/20 0.38
KCNQ3 O43525 2/20 0.38
KCNQ2 O43526 2/20 0.38
KCNE1 P15382 2/20 0.38
KCNQ1 P51787 2/20 0.38
KCNQ5 Q9NR82 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
ADORA1 P30542 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3944917 0.94 BACE1 (0.41) KCNK3KCNK9MAPTNPC1RAB9A
SCHEMBL3944601 0.89 KCNK3 (0.44) KCNK3NPC1RAB9AKMT2AMEN1
SCHEMBL3951861 0.89 GRM4 (0.41) KCNK3KCNK9MAPTNPC1RAB9A
SCHEMBL4154763 0.87 KCNK3 (0.41) KCNK3KCNK9GRM5MAPTBACE1
SCHEMBL3952707 0.87 KCNK3 (0.41) KCNK3KCNK9RAB9ABACE1KMT2A
SCHEMBL3944465 0.85 KCNK3 (0.44) KCNK3KCNK9MAPTTP53BACE1
SCHEMBL3951123 0.85 BACE1 (0.41) NPC1RAB9ABACE1KMT2AMEN1
SCHEMBL3951875 0.85 MAPT (0.42) KCNK3KCNK9MAPTNPC1RAB9A
SCHEMBL3952248 0.84 BACE1 (0.40) BACE1ALDH1A1
SCHEMBL3951984 0.83 SMN1; SMN2 (0.38) KCNK3KCNK9MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed