SCHEMBL3944682

SCHEMBL3944682

CC(=O)c1ccc(-c2c(OC(=O)NCCN3CCOCC3)[nH]c3ccc(NS(=O)(=O)c4ccc(C(C)(C)C)cc4)cc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
CD274 Q9NZQ7 2/20 0.42
POLB P06746 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
BRD4 O60885 1/20 0.40
MMP12 P39900 1/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
EPHX2 P34913 1/20 0.38
SERPINE1 P05121 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3952225 0.93 ALDH1A1 (0.44) ALDH1A1MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL3944430 0.93 ALDH1A1 (0.46) ALDH1A1MEN1MAPTKMT2ACYP1A2
SCHEMBL3943786 0.92 EPHX2 (0.47) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL3941985 0.92 ALDH1A1 (0.46) ALDH1A1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL3953107 0.91 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3950137 0.91 CD274 (0.43) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3949764 0.90 L3MBTL1 (0.43) ALDH1A1MEN1MAPTKMT2ACYP1A2
SCHEMBL3943388 0.89 ALDH1A1 (0.41) ALDH1A1MEN1MAPTKMT2ACYP1A2
SCHEMBL3946197 0.89 ALDH1A1 (0.42) ALDH1A1MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL3942066 0.89 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802572-B1 INDOL DERIVATIVES AS INHIBITORS OF SOLUBLE ADENYLYL CYCLASE BAYER SCHERING PHARMA AG (DE) 2009-04-22 EP claimed
EP-1802572-B1 INDOL DERIVATIVES AS INHIBITORS OF SOLUBLE ADENYLYL CYCLASE BAYER SCHERING PHARMA AG (DE) 2009-04-22 EP disclosed