SCHEMBL3945147

SCHEMBL3945147

CN(CC(O)c1ccc(O)c(O)c1)C(=O)Oc1cnc(N(C)Cc2ccccc2)nc1-c1ccccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSPO P30536 4/20 0.37
CASR P41180 3/20 0.37
PDK1 Q15118 2/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
LMNA P02545 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CCNE2 O96020 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ADRB2 P07550 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3951648 0.91 TSPO (0.37) TSPOCASRPDK1TP53
SCHEMBL3950139 0.91 CASR (0.37) CASRLMNACYP1A2CYP3A4CCNE2
SCHEMBL3951753 0.82 CASR (0.37) CASRMEN1KMT2AKDM4EMAPT
SCHEMBL4036518 0.82 CASR (0.40) CASRPDK1NPSR1MEN1KMT2A
SCHEMBL3943392 0.82 ITGB1 (0.38) CASRPDK1
SCHEMBL3942436 0.81 CASR (0.42) CASRPDK1KDM4ERXFP1
SCHEMBL3945206 0.81 CASR (0.37) CASRPDK1HTTMEN1KMT2A
SCHEMBL3945373 0.81 CASR (0.37) CASRPDK1MEN1KMT2ATP53
SCHEMBL3942465 0.81 CASR (0.41) CASRPDK1PDK2PDK3PDK4
SCHEMBL3947316 0.80 CASR (0.41) CASRPDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed