SCHEMBL3947754

SCHEMBL3947754

CC(C)(C)[N+]1(C(=O)[O-])C[C@H](NS(=O)(=O)c2cc(Br)ccc2Br)C[C@@H]1CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.42
CTSS P25774 2/20 0.42
CTSK P43235 2/20 0.42
CTSC P53634 1/20 0.42
CTSB P07858 1/20 0.37
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MMP1 P03956 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP14 P50281 1/20 0.34
ADAM17 P78536 1/20 0.34
BRD4 O60885 8/20 0.33
RORC P51449 1/20 0.33
MAPT P10636 1/20 0.33
HTR1A P08908 1/20 0.33
HTR7 P34969 1/20 0.33
LPAR2 Q9HBW0 1/20 0.32
APAF1 O14727 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3947518 0.84 MMP2 (0.36) ALDH1A1MMP2MMP9BRD4RORC
SCHEMBL3949052 0.84 CTSL (0.46) CTSLCTSSCTSKCTSCCTSB
SCHEMBL3948515 0.83 CTSL (0.45) CTSLCTSSCTSKCTSCCTSB
SCHEMBL3954902 0.82 KMT2A (0.47) CTSLCTSSCTSKCTSCCTSB
SCHEMBL3951319 0.81 CTSL (0.44) CTSLCTSSCTSKCTSCCTSB
SCHEMBL3949447 0.81 CTSL (0.41) CTSLCTSSCTSKCTSCCTSB
SCHEMBL3954226 0.80 CTSL (0.40) CTSLCTSSCTSKCTSCCTSB
SCHEMBL3950831 0.80 CTSL (0.43) CTSLCTSSCTSKCTSCCTSB
SCHEMBL3955669 0.80 ALDH1A1 (0.44) CTSLCTSSCTSKCTSCCTSB
SCHEMBL3944081 0.79 CTSL (0.39) CTSLCTSSCTSKCTSCCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026197-A1 NOVEL CATHEPSIN C INHIBITORS AND THEIR USE GLAXO GROUP LIMITED (GB) 2009-02-26 WO disclosed