SCHEMBL3949183

SCHEMBL3949183

CC(C)c1nc(Cl)c2ccccc2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
METAP1 P53582 1/20 0.45
NPSR1 Q6W5P4 3/20 0.44
RXFP1 Q9HBX9 3/20 0.44
PRNP P04156 2/20 0.44
TSHR P16473 2/20 0.44
USP2 O75604 1/20 0.44
AURKA O14965 1/20 0.44
AURKB Q96GD4 1/20 0.44
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPT P10636 3/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835430 0.82 PDE4A (0.45) MAOAMAOBMETAP1RXFP1PRNP
SCHEMBL13158216 0.81 MAOA (0.47) MAOAMAOBMETAP1TSHRPDE4A
SCHEMBL11735484 0.78 NPSR1 (0.46) MAOAMAOBNPSR1RXFP1PRNP
SCHEMBL13548854 0.78 GPR3 (0.55) NPSR1RXFP1PRNPTSHRUSP2
SCHEMBL19685360 0.77 PRNP (0.48) NPSR1RXFP1PRNPTSHRUSP2
SCHEMBL4753647 0.77 DCPS (0.57) MAOANPSR1RXFP1PRNPTSHR
SCHEMBL31391449 0.77 RXFP1 (0.44) MAOAMAOBNPSR1RXFP1PRNP
SCHEMBL20152506 0.76 ADORA2A (0.55) NPSR1ALDH1A1MAPTL3MBTL1KMT2A
SCHEMBL856788 0.75 TDP1 (0.54) MAOAMAOBMETAP1NPSR1RXFP1
SCHEMBL29461212 0.75 TDP1 (0.54) MAOAMAOBMETAP1NPSR1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029617-A1 DIARYLAMINE-SUBSTITUTED QUINOLONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed