SCHEMBL3950341

SCHEMBL3950341

Cc1ccnc2[nH]c(CC(C)C)nc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
MAPK8 P45983 2/20 0.33
GSK3A P49840 2/20 0.33
CDK5 Q00535 2/20 0.33
AURKA O14965 1/20 0.33
DAPK3 O43293 1/20 0.33
JAK2 O60674 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
ABL1 P00519 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3952081 0.83 GSK3B (0.38) GSK3BKDM4EMAPTPDE3BPDE3A
SCHEMBL4370028 0.81 ADORA1 (0.41) GSK3BADORA3ADORA2AADORA1MAPK8
SCHEMBL3954959 0.80 GSK3B (0.36) GSK3BKDM4EMAPTPDE3BPDE3A
SCHEMBL28836229 0.80 CCR1 (0.34) GSK3BMAPK8GSK3ACDK5CCR1
SCHEMBL7832083 0.80 KDM4E (0.36) GSK3BKDM4EGSK3ACDK5CCR1
SCHEMBL6317646 0.79 LRRK2 (0.33) MAPTDYRK1ALRRK2CCR1CCR5
Hydrochloric Acid SCHEMBL28836198 0.79 CYP1A2 (0.35) GSK3BMAPK8GSK3ACDK5CCR1
SCHEMBL4370037 0.79 NOS2 (0.41) GSK3BKDM4EPDE3BPDE3AMAPK8
SCHEMBL8875881 0.76 GSK3B (0.44) GSK3BMAPK8GSK3ACDK5MAPK9
SCHEMBL8214129 0.75 CCNB2 (0.40) GSK3BGSK3APDE9APARP14CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed