SCHEMBL3952103

SCHEMBL3952103

c1cnn2cc(C3CCC3)nc2n1

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3954500 0.74 RBP4 (0.39) PDE10AALDH1A1
SCHEMBL17227450 0.70 PDE10A (0.33) PDE10A
SCHEMBL7224641 0.69 KDM4E (0.33) ALDH1A1
SCHEMBL3951474 0.69 GSK3A (0.36) PDE10A
SCHEMBL15767503 0.67 ALDH1A1 (0.51) ALDH1A1
SCHEMBL16283746 0.66 PDE10A (0.58) PDE10A
SCHEMBL4478891 0.66 ALDH1A1 (0.34) PDE10AALDH1A1
SCHEMBL31579337 0.64 CNR2 (0.34) ALDH1A1TSHR
SCHEMBL10797169 0.64 RAB9A (0.64) PDE10AALDH1A1TSHR
SCHEMBL3951531 0.63 KDM5B (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029625-A1 4- [HETEROCYCLYL-METHYL] -8-FLUORO-QUINOLIN-2-ONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed
WO-2009029625-A1 4- [HETEROCYCLYL-METHYL] -8-FLUORO-QUINOLIN-2-ONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed