SCHEMBL3953151

SCHEMBL3953151

COc1ccc2[nH]c(C(=O)O)c(CCO)c2c1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.79
ALDH1A1 P00352 5/20 0.79
HPGD P15428 3/20 0.79
HSD17B10 Q99714 2/20 0.79
POLB P06746 2/20 0.72
MDM2 Q00987 1/20 0.72
GPR17 Q13304 1/20 0.63
MEN1 O00255 3/20 0.60
KMT2A Q03164 3/20 0.60
AKR1C2 P52895 1/20 0.56
MAPT P10636 3/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
NQO2 P16083 1/20 0.54
GAA P10253 3/20 0.53
GSK3A P49840 1/20 0.53
GSK3B P49841 1/20 0.53
GFER P55789 1/20 0.53
CDK5 Q00535 1/20 0.53
CDK5R1 Q15078 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3036074 0.86 KDM4E (0.74) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL9127829 0.86 KDM4E (0.86) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL1345727 0.86 KDM4E (0.73) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL29628842 0.85 KDM4E (0.76) KDM4EALDH1A1HPGDHSD17B10POLB
Hydrochloric Acid SCHEMBL1343869 0.85 ALDH1A1 (0.72) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL15428037 0.84 KDM4E (1.00) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL6703468 0.83 KDM4E (0.69) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL3953976 0.82 HTR6 (0.58) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL4231080 0.80 HTR1D (0.74) KDM4EALDH1A1HSD17B10POLBMEN1
SCHEMBL29201304 0.80 ALDH1A1 (0.65) KDM4EALDH1A1HPGDHSD17B10POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103130705-B Benzo five-membered unsaturated heterocycle compound or its pharmaceutical salts and preparation method thereof, pharmaceutical composition and application thereof INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-04-20 CN disclosed
WO-2009097515-A2 [A]-FUSED INDOLE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2009-08-06 WO disclosed