SCHEMBL3953252

SCHEMBL3953252

FC(F)(F)CCNc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
MAPT P10636 1/20 0.58
L3MBTL1 Q9Y468 2/20 0.50
PTPN1 P18031 1/20 0.39
PTPRZ1 P23471 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
HSD17B10 Q99714 2/20 0.38
CTSD P07339 1/20 0.38
CA12 O43570 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
HDAC3 O15379 1/20 0.37
DRD4 P21917 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
ALOX12 P18054 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28241519 0.80 ALDH1A1 (0.44) ALDH1A1MAPTL3MBTL1TDP1CTSD
SCHEMBL4762870 0.79 MAPT (0.56) ALDH1A1MAPTL3MBTL1HRH3TSHR
SCHEMBL232188 0.79 MAPT (0.78) ALDH1A1MAPTL3MBTL1HRH3TDP1
SCHEMBL549076 0.78 ALDH1A1 (0.54) ALDH1A1MAPTL3MBTL1PTPN1PTPRZ1
SCHEMBL5417854 0.77 APP (0.46) ALDH1A1MAPTL3MBTL1TDP1MAOA
SCHEMBL6416019 0.76 MAPT (0.74) ALDH1A1MAPTL3MBTL1HRH3TDP1
SCHEMBL1562142 0.76 MAPT (0.74) ALDH1A1MAPTL3MBTL1HRH3TDP1
SCHEMBL9572889 0.76 MAPT (0.52) ALDH1A1MAPTL3MBTL1HRH3CA12
SCHEMBL17404465 0.76 PTGS1 (0.59) ALDH1A1CA12CA2CA9PTGS1
SCHEMBL566062 0.75 ALDH1A1 (0.64) ALDH1A1MAPTL3MBTL1HRH3TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078019-A2 PURINES AS PKC-THETA INHIBITORS N.V. Organon (NL) 2009-07-15 EP disclosed
WO-2008051826-A2 PURINES AS PKC-THETA INHIBITORS N.V. ORGANON (NL) 2008-05-02 WO disclosed