SCHEMBL3954017

SCHEMBL3954017

CN(CCN(C)C(=O)O)Cc1ccc(C(=O)NN(c2nc(C#N)ncc2Cl)C2CCCC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 7/20 0.41
CTSL P07711 6/20 0.41
CTSS P25774 6/20 0.41
CTSB P07858 1/20 0.41
SIGMAR1 Q99720 5/20 0.36
TMEM97 Q5BJF2 4/20 0.36
F10 P00742 3/20 0.35
ITK Q08881 1/20 0.33
HIF1A Q16665 1/20 0.33
EPAS1 Q99814 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3959334 0.95 CTSL (0.38) CTSKCTSLCTSSCTSBSIGMAR1
SCHEMBL3168819 0.92 CTSK (0.42) CTSKCTSLCTSSCTSBSIGMAR1
SCHEMBL3165918 0.92 CTSK (0.42) CTSKCTSLCTSSCTSBSIGMAR1
SCHEMBL3166608 0.90 CTSS (0.47) CTSKCTSLCTSSCTSBSIGMAR1
SCHEMBL3166033 0.90 CTSK (0.41) CTSKCTSLCTSSCTSBSIGMAR1
SCHEMBL3170053 0.90 CTSL (0.38) CTSKCTSLCTSSCTSBSIGMAR1
SCHEMBL3176722 0.90 CTSK (0.43) CTSKCTSLCTSSCTSBF10
SCHEMBL3174539 0.89 CTSL (0.47) CTSKCTSLCTSSCTSBSIGMAR1
SCHEMBL3170065 0.89 CTSL (0.38) CTSKCTSLCTSSCTSBSIGMAR1
SCHEMBL3165113 0.89 CTSS (0.46) CTSKCTSLCTSSCTSBSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2077841-A1 NOVEL SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS Glaxo Group Limited (GB) 2009-07-15 EP claimed
WO-2008052934-A1 NOVEL SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2008-05-08 WO claimed