SCHEMBL3957007

SCHEMBL3957007

CC(C)(C)OC(=O)NCC(O)CNCCNC(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
GAA P10253 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.41
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
ADRB2 P07550 1/20 0.38
HTR1A P08908 1/20 0.38
EPHX1 P07099 1/20 0.38
SYK P43405 1/20 0.37
CTSK P43235 5/20 0.36
CTSS P25774 3/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
MALT1 Q9UDY8 1/20 0.36
CA12 O43570 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
SERPINE1 P05121 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3013440 0.92 MEN1 (0.49) MEN1GAAKMT2ATDP1MAOA
SCHEMBL12475162 0.87 MEN1 (0.49) MEN1GAAKMT2ATDP1MAOA
SCHEMBL30299043 0.86 MAOA (0.53) MEN1GAAKMT2ATDP1MAOA
SCHEMBL13960156 0.85 MEN1 (0.46) MEN1GAAKMT2ATDP1MAOA
SCHEMBL16379307 0.85 MEN1 (0.46) MEN1GAAKMT2ATDP1MAOA
SCHEMBL570033 0.83 MEN1 (0.50) MEN1GAAKMT2ATDP1MAOA
SCHEMBL13959822 0.83 MEN1 (0.54) MEN1GAAKMT2ATDP1MAOA
SCHEMBL18614971 0.82 MEN1 (0.54) MEN1GAAKMT2ATDP1MAOA
SCHEMBL3025341 0.82 MAOA (0.44) MEN1GAAKMT2ATDP1MAOA
SCHEMBL1760969 0.80 MEN1 (0.59) MEN1GAAKMT2ATDP1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866291-B1 ANTIBACTERIAL AMIDE MACROCYCLES VI AICURIS GMBH & CO KG (DE) 2009-07-15 EP disclosed
EP-1866291-A1 ANTIBACTERIAL AMIDE MACROCYCLES VI AiCuris GmbH & Co. KG (DE) 2007-12-19 EP disclosed
WO-2006103009-A1 ANTIBACTERIAL AMIDE MACROCYCLES VI AICURIS GMBH & CO. KG (DE) 2006-10-05 WO disclosed