SCHEMBL3958263

SCHEMBL3958263

COc1ccc(C(C)Cc2ccccc2)cc1N

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
PDE4A P27815 2/20 0.43
ALDH1A1 P00352 4/20 0.42
CYP3A4 P08684 2/20 0.42
ADRA2B P18089 1/20 0.42
PTGS1 P23219 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTR2A P28223 1/20 0.42
CYP2C19 P33261 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3958267 0.85 GAA (0.56) GAAPDE4AALDH1A1CYP3A4ADRA2B
Ammonia Solution, Strong SCHEMBL8976449 0.84 PDE4A (0.51) PDE4ATDP1MAPTKMT2A
SCHEMBL11572304 0.83 GAA (0.43) GAAPDE4AALDH1A1CYP3A4TDP1
SCHEMBL19478537 0.79 ALDH1A1 (0.59) GAAPDE4AALDH1A1CYP3A4TDP1
SCHEMBL11584591 0.78 ALDH1A1 (0.63) GAAALDH1A1MEN1MAPTKMT2A
Fumaric Acid SCHEMBL8866086 0.75 CA1 (0.49) PDE4AALDH1A1CYP3A4CYP2C19KMT2A
SCHEMBL12089851 0.75 ALDH1A1 (0.55) GAAALDH1A1CYP3A4ADRA2BPTGS1
SCHEMBL20693253 0.74 TUBB4A (0.41) GAAHTR2A
SCHEMBL31480917 0.74 ALDH1A1 (0.46) GAAALDH1A1CYP3A4ADRA2BPTGS1
SCHEMBL28344005 0.74 ALDH1A1 (0.59) ALDH1A1CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076497-A1 AMINOMETHYL-4-IMIDAZOLES F. Hoffmann-Roche AG (CH) 2009-07-08 EP disclosed
WO-2008046757-A1 AMINOMETHYL-4-IMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2008-04-24 WO disclosed