SCHEMBL3958267

SCHEMBL3958267

COc1ccc(CC(C)c2ccccc2)cc1N

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.56
ALOX15 P16050 1/20 0.43
ALOX12 P18054 1/20 0.43
ALDH1A1 P00352 4/20 0.42
LMNA P02545 1/20 0.42
CYP3A4 P08684 1/20 0.42
LDHA P00338 1/20 0.42
PDE4A P27815 1/20 0.42
ADRA2B P18089 1/20 0.42
PTGS1 P23219 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
KMT2A Q03164 2/20 0.41
NR3C2 P08235 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3958263 0.85 GAA (0.47) GAAALDH1A1CYP3A4PDE4AADRA2B
SCHEMBL27183403 0.82 ALOX15 (0.67) GAAALOX15ALOX12LMNACYP3A4
SCHEMBL11584588 0.78 ALDH1A1 (0.50) GAAALOX15ALOX12ALDH1A1LMNA
SCHEMBL14276990 0.76 SKP2 (0.45) ALDH1A1CYP3A4TDP1SIGMAR1NR3C2
Bromide SCHEMBL6837017 0.76 GAA (0.56) GAAALDH1A1LMNACYP3A4LDHA
SCHEMBL27205449 0.76 GAA (0.65) GAA
SCHEMBL9069704 0.74 ESR1 (0.61) SIGMAR1
SCHEMBL4603238 0.74 MEN1 (0.59) ALDH1A1LDHASIGMAR1KMT2AMEN1
SCHEMBL4603241 0.74 MEN1 (0.59) ALDH1A1LDHASIGMAR1KMT2AMEN1
SCHEMBL8732205 0.73 TAAR1 (0.52) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076497-A1 AMINOMETHYL-4-IMIDAZOLES F. Hoffmann-Roche AG (CH) 2009-07-08 EP disclosed
WO-2008046757-A1 AMINOMETHYL-4-IMIDAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2008-04-24 WO disclosed