SCHEMBL3958356

SCHEMBL3958356

CC(CC(=O)Nc1nccnc1N)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
TLR7 Q9NYK1 2/20 0.33
SMN1; SMN2 Q16637 3/20 0.32
PRKCI P41743 5/20 0.31
SHMT2 P34897 1/20 0.31
ATR Q13535 1/20 0.31
LMNA P02545 1/20 0.30
PTPN1 P18031 2/20 0.30
AAK1 Q2M2I8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13905270 1.00 ALDH1A1 (0.33) ALDH1A1TLR7SMN1; SMN2PRKCISHMT2
SCHEMBL3950119 0.85 TLR7 (0.34) ALDH1A1TLR7PRKCISHMT2ATR
SCHEMBL28162119 0.72 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2PRKCISHMT2ATR
SCHEMBL29200836 0.69 L3MBTL1 (0.41) ALDH1A1PRKCIATR
SCHEMBL3949363 0.68 POLB (0.47) ALDH1A1SMN1; SMN2LMNA
SCHEMBL19597568 0.67 ATR (0.44) ALDH1A1TLR7PRKCISHMT2ATR
SCHEMBL3949001 0.67 EPHX2 (0.46) SMN1; SMN2AAK1
SCHEMBL13560302 0.65 ECE1 (0.37)
SCHEMBL28389860 0.65 MAP4K4 (0.43) PRKCIATR
SCHEMBL30281178 0.65 SMN1; SMN2 (0.40) ALDH1A1TLR7SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed