SCHEMBL3963250

SCHEMBL3963250

Cc1cccc(C(=O)C2CCCN(C(=O)O)C2)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.56
RHOA P61586 1/20 0.54
MEN1 O00255 7/20 0.50
KMT2A Q03164 7/20 0.50
ALDH1A1 P00352 3/20 0.50
KDM2B Q8NHM5 2/20 0.50
POLB P06746 2/20 0.50
MAPK1 P28482 1/20 0.50
HSD11B1 P28845 1/20 0.50
FAAH O00519 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MAPT P10636 1/20 0.50
MGLL Q99685 1/20 0.50
PKM P14618 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21926317 0.90 HPGD (0.60) HPGDRHOAMEN1KMT2AALDH1A1
SCHEMBL17913800 0.85 MEN1 (0.68) MEN1KMT2AALDH1A1KDM2BMAPK1
SCHEMBL3723522 0.84 ALDH1A1 (0.61) MEN1KMT2AALDH1A1KDM2BMAPK1
SCHEMBL3324359 0.84 KDM2B (0.69) ALDH1A1KDM2BL3MBTL1MGLL
SCHEMBL4082779 0.84 ALDH1A1 (0.61) HPGDMEN1KMT2AALDH1A1KDM2B
SCHEMBL3966828 0.84 KDM2B (0.69) ALDH1A1KDM2BL3MBTL1MGLL
SCHEMBL16447329 0.83 MGLL (0.64) HPGDMEN1KMT2AALDH1A1HSD11B1
Hydrochloric Acid SCHEMBL6998897 0.83 ALDH1A1 (0.60) MEN1KMT2AALDH1A1KDM2BMAPK1
SCHEMBL2328924 0.83 USP30 (0.53) HPGDRHOAMEN1KMT2AALDH1A1
SCHEMBL2328921 0.83 USP30 (0.53) HPGDRHOAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101356156-B Aspartic protease inhibitors VITAE PHARMACEUTICALS INC 2012-12-05 CN disclosed
EP-2081927-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2009-07-29 EP disclosed
CN-101356156-A Aspartic protease inhibitors VITAE PHARMACEUTICALS INC (US) 2009-01-28 CN disclosed
EP-1966139-A1 ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2008-09-10 EP disclosed
WO-2008036216-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2008-03-27 WO disclosed
WO-2007070201-A1 ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-06-21 WO disclosed