SCHEMBL4082779

SCHEMBL4082779

O=C(c1cccc(F)c1)C1CCCN(C(=O)O)C1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
MEN1 O00255 3/20 0.61
KMT2A Q03164 3/20 0.61
HSD11B1 P28845 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
HTT P42858 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.52
KDM4E B2RXH2 1/20 0.51
HPGD P15428 1/20 0.51
MGLL Q99685 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
KDM2B Q8NHM5 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3723522 0.84 ALDH1A1 (0.61) ALDH1A1MEN1KMT2AL3MBTL1CYP2C9
SCHEMBL3324359 0.84 KDM2B (0.69) ALDH1A1KDM4EMGLLL3MBTL1KDM2B
SCHEMBL3963250 0.84 HPGD (0.56) ALDH1A1MEN1KMT2AHSD11B1HPGD
SCHEMBL3966828 0.84 KDM2B (0.69) ALDH1A1KDM4EMGLLL3MBTL1KDM2B
SCHEMBL3895577 0.83 HSD11B1 (0.69) MEN1KMT2AHSD11B1TDP1MGLL
Hydrochloric Acid SCHEMBL6998897 0.83 ALDH1A1 (0.60) ALDH1A1MEN1KMT2AL3MBTL1CYP2C9
SCHEMBL5476575 0.83 ALDH1A1 (0.67) ALDH1A1MEN1KMT2A
SCHEMBL5476573 0.83 ALDH1A1 (0.67) ALDH1A1MEN1KMT2A
SCHEMBL969182 0.82 ALDH1A1 (0.59) ALDH1A1MEN1KMT2A
SCHEMBL5475032 0.82 ALDH1A1 (0.59) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101356156-B Aspartic protease inhibitors VITAE PHARMACEUTICALS INC 2012-12-05 CN disclosed
EP-2074108-A1 RENIN INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2009-07-01 EP disclosed
CN-101356156-A Aspartic protease inhibitors VITAE PHARMACEUTICALS INC (US) 2009-01-28 CN disclosed
EP-1966139-A1 ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2008-09-10 EP disclosed
WO-2008036247-A1 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2008-03-27 WO disclosed
WO-2007070201-A1 ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-06-21 WO disclosed