SCHEMBL3970388

SCHEMBL3970388

CCOc1cc(CN(c2cc(C#N)ccn2)C2CCNCC2)cc(OCC)c1F

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 6/20 0.39
SLC6A4 P31645 6/20 0.39
SLC6A3 Q01959 5/20 0.39
HTR6 P50406 2/20 0.38
HCRTR1 O43613 6/20 0.37
HCRTR2 O43614 6/20 0.37
IKBKB O14920 1/20 0.36
NR3C2 P08235 2/20 0.36
NR3C1 P04150 1/20 0.36
PGR P06401 1/20 0.36
AR P10275 1/20 0.36
NOS3 P29474 2/20 0.34
NOS1 P29475 2/20 0.34
NOS2 P35228 2/20 0.34
MAP3K12 Q12852 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973243 0.88 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3HTR6HCRTR1
SCHEMBL3973780 0.87 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3HTR6HCRTR1
SCHEMBL3972380 0.86 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3HTR6IKBKB
SCHEMBL3972445 0.82 SSTR5 (0.40) SLC6A2SLC6A4SLC6A3
SCHEMBL3969984 0.79 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL4594518 0.79 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3HTR6IKBKB
SCHEMBL3972485 0.77 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3HTR6IKBKB
SCHEMBL3973733 0.77 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3HTR6IKBKB
SCHEMBL3972502 0.77 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3HTR6IKBKB
SCHEMBL3973888 0.77 IKBKB (0.40) SLC6A2SLC6A4SLC6A3HTR6IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP claimed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO claimed
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed