SCHEMBL3969984

SCHEMBL3969984

CC(C)Oc1cc(CN(c2cc(C#N)ccn2)C2CCNCC2)cc(OC(C)C)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.44
SLC6A4 P31645 12/20 0.44
SLC6A3 Q01959 8/20 0.44
MAP3K12 Q12852 1/20 0.39
NOS1 P29475 2/20 0.36
NOS2 P35228 2/20 0.36
NOS3 P29474 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.35
HTR2A P28223 1/20 0.35
HTR3A P46098 1/20 0.34
KCNH2 Q12809 1/20 0.34
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973401 0.86 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3NOS1NOS2
SCHEMBL3974287 0.82 IRAK4 (0.42) SLC6A2SLC6A4SLC6A3IRAK4HTR2A
SCHEMBL3970388 0.79 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3MAP3K12NOS1
SCHEMBL4703738 0.78 SLC6A2 (0.48) SLC6A2SLC6A4SLC6A3IRAK4HTR2A
SCHEMBL3973243 0.77 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3NOS1NOS2
SCHEMBL4703851 0.76 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3NOS1NOS2
SCHEMBL3973780 0.76 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3NOS1NOS2
SCHEMBL4259000 0.74 GCK (0.44)
SCHEMBL3938776 0.74 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3HTR2A
SCHEMBL3974019 0.74 MBTPS1 (0.40) SLC6A2SLC6A4SLC6A3IRAK4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP claimed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO claimed
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed