SCHEMBL3973243

SCHEMBL3973243

CCOc1cc(CN(c2cc(C#N)ccn2)C2CCNCC2)ccc1C

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 7/20 0.41
SLC6A4 P31645 7/20 0.41
SLC6A3 Q01959 6/20 0.41
HTR6 P50406 1/20 0.40
NR3C2 P08235 3/20 0.38
NR3C1 P04150 2/20 0.38
PGR P06401 2/20 0.38
AR P10275 2/20 0.38
HCRTR1 O43613 5/20 0.37
HCRTR2 O43614 5/20 0.37
IKBKB O14920 1/20 0.36
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
KCNH2 Q12809 1/20 0.33
KDM1A O60341 1/20 0.33
TACR1 P25103 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973780 0.90 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3HTR6NR3C2
SCHEMBL3970388 0.88 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3HTR6NR3C2
SCHEMBL3972421 0.86 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3HTR6NR3C2
SCHEMBL3971762 0.83 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3IKBKBKCNH2
SCHEMBL3939276 0.78 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3HTR6IKBKB
SCHEMBL3969984 0.77 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3HTR6NOS3
SCHEMBL3976469 0.77 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3HTR6IKBKB
SCHEMBL3972485 0.77 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3HTR6IKBKB
SCHEMBL3970914 0.77 IKBKB (0.41) SLC6A2SLC6A4SLC6A3HTR6IKBKB
SCHEMBL3973911 0.77 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3NR3C2NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP claimed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO claimed
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed