SCHEMBL3972873

SCHEMBL3972873

CCOc1cc(CN(c2ccc(C(N)=O)cn2)C2CCNCC2)ccc1F

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.37
SLC6A5 Q9Y345 1/20 0.37
KCNH2 Q12809 3/20 0.37
SLC6A2 P23975 3/20 0.37
SLC6A4 P31645 3/20 0.37
SLC6A3 Q01959 3/20 0.37
TACR1 P25103 4/20 0.36
SSTR5 P35346 2/20 0.34
MAPK1 P28482 1/20 0.34
REN P00797 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3979779 0.92 RXRA (0.41) SLC6A9SLC6A5KCNH2SLC6A2SLC6A4
SCHEMBL3973958 0.91 SSTR5 (0.40) KCNH2SLC6A2SLC6A4SLC6A3TACR1
SCHEMBL3977612 0.90 SLC6A2 (0.37) KCNH2SLC6A2SLC6A4SLC6A3TACR1
SCHEMBL3972925 0.90 MAPK1 (0.44) KCNH2SLC6A2SLC6A4SLC6A3MAPK1
SCHEMBL3971901 0.90 SSTR5 (0.43) KCNH2SLC6A2SLC6A4SLC6A3TACR1
SCHEMBL3973812 0.89 SSTR5 (0.38) KCNH2SLC6A2SLC6A4SLC6A3TACR1
SCHEMBL3971524 0.88 MAPK1 (0.36) KCNH2SLC6A2SLC6A4SLC6A3TACR1
SCHEMBL3977954 0.87 TACR1 (0.37) KCNH2SLC6A2SLC6A4SLC6A3TACR1
SCHEMBL4705165 0.87 SLC6A2 (0.41) SLC6A9SLC6A5KCNH2SLC6A2SLC6A4
SCHEMBL3977915 0.84 PARP10 (0.39) KCNH2SLC6A2SLC6A4SLC6A3TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP claimed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO claimed
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed