SCHEMBL3979779

SCHEMBL3979779

CCOc1cc(CN(c2ccc(C(=O)O)cn2)C2CCNCC2)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RXRA P19793 11/20 0.41
PPARG P37231 1/20 0.39
SLC6A9 P48067 2/20 0.38
SLC6A5 Q9Y345 1/20 0.38
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
KCNH2 Q12809 2/20 0.37
HCAR3 P49019 2/20 0.37
MAPT P10636 1/20 0.37
TACR1 P25103 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3972873 0.92 SLC6A9 (0.37) SLC6A9SLC6A5SLC6A2SLC6A4SLC6A3
SCHEMBL3978560 0.91 RXRA (0.42) RXRAPPARGHCAR3MAPT
SCHEMBL3973372 0.90 RXRA (0.41) RXRAPPARGSLC6A2SLC6A4SLC6A3
SCHEMBL3973033 0.90 SSTR5 (0.42) RXRAPPARGSLC6A2SLC6A4SLC6A3
SCHEMBL3973856 0.89 L3MBTL1 (0.47) RXRAPPARGMAPT
SCHEMBL3977983 0.89 SSTR5 (0.41) RXRAPPARGSLC6A2SLC6A4SLC6A3
SCHEMBL3972951 0.87 RXRA (0.42) RXRAPPARGHCAR3MAPTTACR1
SCHEMBL3973405 0.84 RXRA (0.42) RXRAPPARGSLC6A2SLC6A4SLC6A3
SCHEMBL3972485 0.83 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3
SCHEMBL3973958 0.83 SSTR5 (0.40) RXRASLC6A2SLC6A4SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP claimed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO claimed
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed