SCHEMBL3973152

SCHEMBL3973152

COC(=O)[C@@H](N)Cc1ccc(-c2ccc(Oc3ccccc3)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 1/20 0.52
ACACB O00763 4/20 0.50
ACACA Q13085 3/20 0.50
LTA4H P09960 1/20 0.50
SCN9A Q15858 1/20 0.49
PPARG P37231 7/20 0.49
PPARA Q07869 7/20 0.49
PPARD Q03181 2/20 0.49
MMP12 P39900 1/20 0.48
MMP13 P45452 1/20 0.48
FFAR1 O14842 1/20 0.48
PTGS2 P35354 1/20 0.47
NPY5R Q15761 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973157 1.00 TPH1 (0.52) TPH1ACACBACACALTA4HSCN9A
SCHEMBL29183302 0.96 ACACB (0.53) TPH1ACACBLTA4HPPARGPPARA
SCHEMBL2292317 0.96 ACACB (0.53) TPH1ACACBLTA4HPPARGPPARA
SCHEMBL8255298 0.96 ACACB (0.53) TPH1ACACBLTA4HPPARGPPARA
Hydrochloric Acid SCHEMBL2292315 0.94 PPARG (0.54) TPH1ACACBLTA4HPPARGPPARA
Hydrochloric Acid SCHEMBL2292318 0.94 PPARG (0.54) TPH1ACACBLTA4HPPARGPPARA
SCHEMBL7451018 0.90 SRR (0.54) TPH1ACACBLTA4HPPARGPPARA
SCHEMBL539325 0.90 SRR (0.54) TPH1ACACBLTA4HPPARGPPARA
SCHEMBL539324 0.90 SRR (0.54) TPH1ACACBLTA4HPPARGPPARA
SCHEMBL20240307 0.89 LTA4H (0.53) ACACBACACALTA4HPPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7501538-B2 Aryl and heteroaryl compounds, compositions and methods of use TRANSTECH PHARMA, INC. (US) 2009-03-10 US disclosed
US-20050049310-A1 Aryl and heteroaryl compounds, compositions and methods of use VTVX HOLDINGS I LLC 2005-03-03 US disclosed
WO-2005014532-A1 ARYL AND HETEROARYL COMPOUNDS, COMPOSITIONS AND METHODS OF USE TRANSTECH PHARMA, INC. (US) 2005-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050049310-A1 Aryl and heteroaryl compounds, compositions and methods of use EPOR, HBG2, CYP2F1 TPH1 1389/4885ACACB 1320/4885ACACA 1118/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.