SCHEMBL3973539

SCHEMBL3973539

CCCCCNc1cc(C(=O)O)c(Br)cc1C(N)=O

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CISD1 Q9NZ45 8/20 0.54
KDM6B O15054 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
HCAR3 P49019 1/20 0.41
PLK1 P53350 4/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
CA14 Q9ULX7 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2429407 0.96 CISD1 (0.53) CISD1KDM6BKDM4CHCAR3CA12
SCHEMBL2431511 0.90 CISD1 (0.51) CISD1KDM6BKDM4CHCAR3CA12
SCHEMBL2426202 0.85 CISD1 (0.52) CISD1KDM6BKDM4CHCAR3PLK1
SCHEMBL3979546 0.84 CISD1 (0.51) CISD1KDM6BKDM4CHCAR3PLK1
SCHEMBL1884483 0.82 CISD1 (0.63) CISD1KDM6BKDM4CHCAR3PLK1
SCHEMBL3974778 0.81 CISD1 (0.48) CISD1KDM6BKDM4CHCAR3PLK1
SCHEMBL2422093 0.78 APEX1 (0.36) CISD1CA12CA1CA2CA3
SCHEMBL2425743 0.78 MAPK8 (0.42) CISD1CA12CA1CA2CA3
SCHEMBL2428525 0.78 TSHR (0.46) CISD1KDM6BKDM4CHCAR3CA12
SCHEMBL3141041 0.77 HCAR3 (0.57) CISD1KDM6BKDM4CHCAR3PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed