SCHEMBL3979546

SCHEMBL3979546

CCCCCNc1cc(C(=O)O)c(F)cc1C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CISD1 Q9NZ45 8/20 0.51
KDM6B O15054 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
PLK1 P53350 4/20 0.42
HCAR3 P49019 1/20 0.41
RARB P10826 2/20 0.41
RARA P10276 1/20 0.41
RARG P13631 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2426202 0.85 CISD1 (0.52) CISD1KDM6BKDM4CPLK1HCAR3
SCHEMBL3973539 0.84 CISD1 (0.54) CISD1KDM6BKDM4CPLK1HCAR3
SCHEMBL19665937 0.83 CISD1 (0.43) CISD1PLK1
SCHEMBL3974778 0.83 CISD1 (0.48) CISD1KDM6BKDM4CPLK1HCAR3
SCHEMBL1884483 0.82 CISD1 (0.63) CISD1KDM6BKDM4CPLK1HCAR3
SCHEMBL17363127 0.80 CISD1 (0.56) CISD1KDM6BKDM4CPLK1HCAR3
SCHEMBL2429407 0.80 CISD1 (0.53) CISD1KDM6BKDM4CHCAR3
SCHEMBL3141041 0.77 HCAR3 (0.57) CISD1KDM6BKDM4CPLK1HCAR3
SCHEMBL3973709 0.76 HCAR3 (0.56) CISD1PLK1HCAR3
SCHEMBL2422797 0.75 HCAR3 (0.39) HCAR3RARBRARARARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed