SCHEMBL3973544

SCHEMBL3973544

Cc1cc(C(N)=O)c(NCCCC2CC2)cc1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.39
HSP90AB1 P08238 2/20 0.39
CISD1 Q9NZ45 7/20 0.36
ACP1 P24666 3/20 0.36
LIPC P11150 1/20 0.36
LIPG Q9Y5X9 1/20 0.36
NOTUM Q6P988 1/20 0.35
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
CD38 P28907 1/20 0.34
GUCY1A1 Q02108 1/20 0.34
GUCY1B1 Q02153 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3980322 0.92 HSP90AA1 (0.40) HSP90AA1HSP90AB1CISD1LIPCLIPG
SCHEMBL2430530 0.84 HSP90AA1 (0.48) HSP90AA1HSP90AB1LIPCLIPGNOTUM
SCHEMBL2426202 0.82 CISD1 (0.52) CISD1
SCHEMBL4010874 0.81 GUCY1A1 (0.40) HSP90AA1HSP90AB1CISD1GUCY1A1GUCY1B1
SCHEMBL2431005 0.80 CISD1 (0.49) HSP90AA1HSP90AB1CISD1
SCHEMBL2427599 0.80 ASPH (0.50) HSP90AA1HSP90AB1LIPCLIPGCD38
SCHEMBL2434508 0.78 CISD1 (0.34) HSP90AA1HSP90AB1CISD1CD38GUCY1A1
SCHEMBL3980350 0.76 HSP90AA1 (0.35) HSP90AA1HSP90AB1CISD1CD38
SCHEMBL2422460 0.76 JAK2 (0.40) HSP90AA1HSP90AB1CISD1
SCHEMBL3975516 0.74 RXRB (0.34) HSP90AA1HSP90AB1CISD1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed