SCHEMBL4010874

SCHEMBL4010874

Cc1cc(C(N)=O)c(NCCCC(F)(F)F)cc1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GUCY1A1 Q02108 1/20 0.40
GUCY1B1 Q02153 1/20 0.40
CISD1 Q9NZ45 8/20 0.37
PLK1 P53350 3/20 0.34
KDM4C Q9H3R0 2/20 0.33
BCL2L1 Q07817 1/20 0.33
MCL1 Q07820 1/20 0.33
KDM6B O15054 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
NNMT P40261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2434508 0.92 CISD1 (0.34) GUCY1A1GUCY1B1CISD1HSP90AA1HSP90AB1
SCHEMBL2426202 0.83 CISD1 (0.52) CISD1PLK1KDM4CKDM6B
SCHEMBL3973544 0.81 HSP90AA1 (0.39) GUCY1A1GUCY1B1CISD1HSP90AA1HSP90AB1
SCHEMBL2431005 0.81 CISD1 (0.49) CISD1PLK1KDM4CKDM6BHSP90AA1
SCHEMBL3975516 0.80 RXRB (0.34) CISD1KDM4CHSP90AA1HSP90AB1NNMT
SCHEMBL3980322 0.78 HSP90AA1 (0.40) CISD1KDM4CHSP90AA1HSP90AB1
SCHEMBL4258452 0.78 MEN1 (0.34) CISD1KDM4CKDM6BHSP90AA1HSP90AB1
SCHEMBL2422460 0.77 JAK2 (0.40) CISD1HSP90AA1HSP90AB1NNMT
SCHEMBL2422093 0.76 APEX1 (0.36) CISD1
SCHEMBL2425956 0.75 NNMT (0.37) NNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed