SCHEMBL3974212

SCHEMBL3974212

COC(=O)c1ccc2[nH]cc(CCO)c2c1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.80
GPR84 Q9NQS5 1/20 0.68
CYP2D6 P10635 2/20 0.62
HTR2C P28335 2/20 0.56
HTR1A P08908 3/20 0.56
HTR1D P28221 2/20 0.56
HTR1B P28222 2/20 0.56
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53
HTR7 P34969 2/20 0.53
CYP1A2 P05177 2/20 0.53
HSD17B10 Q99714 2/20 0.53
TSHR P16473 1/20 0.53
HTR5A P47898 1/20 0.53
HTR6 P50406 1/20 0.53
POLB P06746 1/20 0.53
CDK2 P24941 1/20 0.53
ATM Q13315 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MTNR1A P48039 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4349467 0.92 NPC1 (0.68) NPC1GPR84CYP2D6HTR2CHTR1A
SCHEMBL12844152 0.89 GPR84 (0.68) NPC1GPR84CYP2D6HTR2CHTR1A
SCHEMBL2161423 0.89 GPR84 (0.76) NPC1GPR84HTR2CHTR1AHTR1D
SCHEMBL8806861 0.88 GPR84 (0.67) NPC1GPR84CYP2D6HTR2CHTR1A
SCHEMBL27427278 0.88 GPR84 (0.67) NPC1GPR84CYP2D6HTR2CHTR1A
SCHEMBL2534004 0.88 HTR1A (0.73) NPC1GPR84CYP2D6HTR2CHTR1A
SCHEMBL22554662 0.87 GPR84 (0.73) NPC1GPR84HTR2CHTR1AHTR1D
SCHEMBL29871648 0.87 GPR84 (0.87) NPC1GPR84HTR2CHTR1AHTR1D
SCHEMBL28868186 0.85 KMT2A (0.65) NPC1GPR84CYP2D6HTR2CHTR1A
SCHEMBL9263244 0.85 GPR84 (0.64) NPC1GPR84CYP2D6HTR2CHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed