SCHEMBL3974619

SCHEMBL3974619

CC(=O)c1ccc(-c2sc(N)c(C(=O)c3ccccc3)c2-c2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 14/20 0.67
CNR2 P34972 1/20 0.51
GRM6 O15303 2/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49
ADORA2A P29274 9/20 0.45
ADORA2B P29275 9/20 0.45
ADORA3 P0DMS8 6/20 0.45
SRD5A2 P31213 1/20 0.43
RORB Q92753 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3976892 0.93 ADORA1 (0.68) ADORA1CNR2GRM6MEN1ALDH1A1
SCHEMBL4090650 0.92 ADORA1 (0.77) ADORA1CNR2GRM6MEN1ALDH1A1
SCHEMBL4086503 0.91 ADORA1 (0.72) ADORA1CNR2GRM6MEN1ALDH1A1
SCHEMBL4076833 0.89 ADORA1 (0.66) ADORA1CNR2GRM6MEN1ALDH1A1
SCHEMBL4078131 0.88 ADORA1 (0.68) ADORA1CNR2GRM6MEN1ALDH1A1
SCHEMBL3975104 0.84 GRM6 (0.60) ADORA1GRM6MEN1ALDH1A1CYP1A2
SCHEMBL4080808 0.80 ADORA1 (0.75) ADORA1CNR2GRM6MEN1ALDH1A1
SCHEMBL4091366 0.80 ADORA1 (1.00) ADORA1CNR2GRM6MEN1ALDH1A1
SCHEMBL3974618 0.79 ADORA1 (0.44) ADORA1CNR2MEN1ALDH1A1CYP1A2
SCHEMBL3981712 0.78 GRM6 (0.57) ADORA1GRM6MEN1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049362-A1 A1 ADENOSINE RECEPTOR ALLOSTERIC ENHANCERS MONASH UNIVERSITY (AU) 2009-04-23 WO disclosed