SCHEMBL4091366

SCHEMBL4091366

Nc1sc(Br)c(-c2cccc(C(F)(F)F)c2)c1C(=O)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 1.00
CNR2 P34972 3/20 0.57
MAPT P10636 2/20 0.52
ALDH1A1 P00352 2/20 0.52
MEN1 O00255 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
KMT2A Q03164 1/20 0.52
HSD17B10 Q99714 1/20 0.52
RORB Q92753 7/20 0.47
SRD5A2 P31213 1/20 0.45
CNR1 P21554 1/20 0.44
GRM6 O15303 1/20 0.43
CES2 O00748 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4090650 0.87 ADORA1 (0.77) ADORA1CNR2MAPTALDH1A1MEN1
SCHEMBL4080808 0.86 ADORA1 (0.75) ADORA1CNR2MAPTALDH1A1MEN1
SCHEMBL4086503 0.84 ADORA1 (0.72) ADORA1CNR2MAPTALDH1A1MEN1
SCHEMBL3976892 0.81 ADORA1 (0.68) ADORA1CNR2MAPTALDH1A1MEN1
SCHEMBL4078131 0.81 ADORA1 (0.68) ADORA1CNR2MAPTALDH1A1MEN1
SCHEMBL3974619 0.80 ADORA1 (0.67) ADORA1CNR2MAPTALDH1A1MEN1
SCHEMBL4076833 0.79 ADORA1 (0.66) ADORA1CNR2MAPTALDH1A1MEN1
SCHEMBL3976346 0.78 ADORA1 (0.63) ADORA1CNR2MAPTALDH1A1MEN1
SCHEMBL3980569 0.76 ADORA1 (0.61) ADORA1CNR2MAPTALDH1A1MEN1
SCHEMBL4091364 0.72 ADORA1 (0.56) ADORA1CNR2MAPTRORB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049362-A1 A1 ADENOSINE RECEPTOR ALLOSTERIC ENHANCERS MONASH UNIVERSITY (AU) 2009-04-23 WO disclosed