SCHEMBL3974618

SCHEMBL3974618

CC(=O)c1ccc(-c2sc(N)c(-c3ccccc3C=O)c2-c2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.44
CNR2 P34972 2/20 0.38
RORB Q92753 5/20 0.37
GPR52 Q9Y2T5 1/20 0.37
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MAOB P27338 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35
RORC P51449 1/20 0.35
SLC9A1 P19634 1/20 0.35
KIF11 P52732 1/20 0.34
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
IKBKB O14920 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3976889 0.93 ADORA1 (0.46) ADORA1CNR2RORBALDH1A1MEN1
SCHEMBL4090647 0.89 ADORA1 (0.46) ADORA1CNR2RORBALDH1A1MAOB
SCHEMBL4078130 0.86 ADORA1 (0.40) ADORA1RORBMAPTMAOBRORC
SCHEMBL4076829 0.86 RORB (0.41) ADORA1RORBALDH1A1MEN1KMT2A
SCHEMBL3974619 0.79 ADORA1 (0.67) ADORA1CNR2RORBALDH1A1MEN1
SCHEMBL4091364 0.79 ADORA1 (0.56) ADORA1CNR2RORBMAPTMAOB
SCHEMBL4080804 0.79 ADORA1 (0.43) ADORA1CNR2RORBMAPTMAOB
SCHEMBL3975104 0.74 GRM6 (0.60) ADORA1GPR52ALDH1A1MEN1KMT2A
SCHEMBL3976892 0.72 ADORA1 (0.68) ADORA1CNR2RORBALDH1A1MEN1
SCHEMBL4085898 0.72 ADORA1 (0.42) ADORA1CNR2RORBALDH1A1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049362-A1 A1 ADENOSINE RECEPTOR ALLOSTERIC ENHANCERS MONASH UNIVERSITY (AU) 2009-04-23 WO disclosed