SCHEMBL4086503

SCHEMBL4086503

Nc1sc(-c2ccc(C(F)(F)F)cc2)c(-c2cccc(C(F)(F)F)c2)c1C(=O)c1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 14/20 0.72
CNR2 P34972 2/20 0.55
MAPT P10636 2/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
KMT2A Q03164 1/20 0.50
HSD17B10 Q99714 1/20 0.50
GRM6 O15303 1/20 0.50
ADORA2A P29274 9/20 0.47
ADORA2B P29275 9/20 0.47
ADORA3 P0DMS8 6/20 0.47
SRD5A2 P31213 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4090650 0.96 ADORA1 (0.77) ADORA1CNR2MAPTMEN1ALDH1A1
SCHEMBL4078131 0.92 ADORA1 (0.68) ADORA1CNR2MAPTMEN1ALDH1A1
SCHEMBL3974619 0.91 ADORA1 (0.67) ADORA1CNR2MAPTMEN1ALDH1A1
SCHEMBL4076833 0.91 ADORA1 (0.66) ADORA1CNR2MAPTMEN1ALDH1A1
SCHEMBL3976892 0.88 ADORA1 (0.68) ADORA1CNR2MAPTMEN1ALDH1A1
SCHEMBL4091366 0.84 ADORA1 (1.00) ADORA1CNR2MAPTMEN1ALDH1A1
SCHEMBL4080808 0.84 ADORA1 (0.75) ADORA1CNR2MAPTMEN1ALDH1A1
SCHEMBL3980249 0.79 GRM6 (0.73) ADORA1MAPTMEN1ALDH1A1CYP1A2
SCHEMBL3975104 0.75 GRM6 (0.60) ADORA1MAPTMEN1ALDH1A1CYP1A2
SCHEMBL3980569 0.74 ADORA1 (0.61) ADORA1CNR2MAPTMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049362-A1 A1 ADENOSINE RECEPTOR ALLOSTERIC ENHANCERS MONASH UNIVERSITY (AU) 2009-04-23 WO disclosed