SCHEMBL3974848

SCHEMBL3974848

O=C(c1ccc(F)cc1)C1(CO)CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 13/20 0.40
SLC6A4 P31645 13/20 0.40
SLC6A3 Q01959 13/20 0.40
CYP2D6 P10635 11/20 0.39
OPRD1 P41143 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
PTPN1 P18031 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4635894 0.86 OPRD1 (0.44) SLC6A2SLC6A4SLC6A3CYP2D6OPRD1
SCHEMBL229151 0.78 CES2 (0.42) OPRD1CES2CES1PTPN1NPC1
SCHEMBL230343 0.78 CES2 (0.42) SLC6A3OPRD1CES2CES1PTPN1
SCHEMBL414713 0.78 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL227735 0.77 CES2 (0.41) OPRD1CES2CES1PTPN1NPC1
SCHEMBL373783 0.75 HDAC1 (0.42) OPRD1CES2CES1CA1CA2
Bromide SCHEMBL10966858 0.75 OPRD1 (0.40) OPRD1CES2CES1PTPN1NPC1
SCHEMBL9377225 0.72 OPRM1 (0.50) OPRD1
SCHEMBL414984 0.70 SLC6A2 (0.79) SLC6A2SLC6A4SLC6A3CYP2D6NPC1
SCHEMBL413666 0.70 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3CYP2D6OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058306-A1 Heteroaryl-substituted 2-pyridinyl-methylamine derivatives SCHWARZ PHARMA AG (DE) 2009-05-13 EP disclosed