SCHEMBL3974923

SCHEMBL3974923

CCCCOc1cc(C(=O)O)c(C)cc1C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.49
NR1I2 O75469 1/20 0.49
LMNA P02545 1/20 0.49
CHRM2 P08172 1/20 0.49
CYP3A4 P08684 1/20 0.49
ADRA2A P08913 1/20 0.49
MAPT P10636 1/20 0.49
OPRK1 P41145 1/20 0.49
HTR2B P41595 1/20 0.49
SLC6A3 Q01959 1/20 0.49
KMT2A Q03164 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
PTPN11 Q06124 4/20 0.46
TP53 P04637 2/20 0.45
RARB P10826 1/20 0.44
WDR5 P61964 2/20 0.44
S1PR3 Q99500 1/20 0.43
RXRA P19793 1/20 0.43
TSHR P16473 1/20 0.42
PLA2G4B P0C869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13270519 0.87 TP53 (0.52) PTPN11TP53RARBWDR5S1PR3
SCHEMBL2429973 0.87 NNMT (0.41) LMNAMAPTKMT2ARARBALDH1A1
SCHEMBL13299048 0.82 TP53 (0.48) PTPN11TP53RARBPLA2G4B
SCHEMBL18133789 0.81 PTPN11 (0.58) PTPN11TP53S1PR3TSHRPLA2G4B
SCHEMBL26454606 0.79 RXRA (0.47) ADRA2AOPRK1PTPN11TP53RARB
SCHEMBL2424366 0.79 ALDH1A1 (0.50) CYP3A4ALDH1A1HPGD
SCHEMBL8167721 0.79 PTPN11 (0.61) PTPN11TP53S1PR3TSHRPLA2G4B
Hydrochloric Acid SCHEMBL9038246 0.77 PTPN11 (0.60) PTPN11TP53S1PR3TSHRPLA2G4B
SCHEMBL10539639 0.77 PTPN11 (0.64) PTPN11TP53RARBS1PR3TSHR
Hydrochloric Acid SCHEMBL8154036 0.77 PTPN11 (0.60) PTPN11TP53S1PR3TSHRPLA2G4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed