SCHEMBL3976791

SCHEMBL3976791

O=C1c2ccc(Cl)cc2C(=O)N1c1ccccc1N1C(=O)c2ccc(Cl)cc2C1=O

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
S100A4 P26447 2/20 0.50
CYP3A4 P08684 1/20 0.49
NFKB1 P19838 1/20 0.49
PMP22 Q01453 1/20 0.49
ESR1 P03372 3/20 0.47
ESR2 Q92731 2/20 0.47
DNM2 P50570 1/20 0.47
ALDH1A1 P00352 2/20 0.46
APEX1 P27695 1/20 0.46
POLB P06746 1/20 0.46
ALDH2 P05091 1/20 0.45
ALDH3A1 P30838 1/20 0.45
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28407461 0.84 MEN1 (0.42) MEN1KMT2AS100A4CYP3A4NFKB1
SCHEMBL1500602 0.83 MEN1 (0.67) MEN1KMT2AS100A4ESR1ESR2
Isothiocyanate SCHEMBL1548406 0.81 KMT2A (0.48) MEN1KMT2AESR1ESR2ALDH1A1
SCHEMBL5903417 0.80 ESR1 (0.61) MEN1KMT2AESR1ESR2
SCHEMBL2884641 0.80 MEN1 (0.62) MEN1KMT2AS100A4ESR1ALDH1A1
SCHEMBL1735121 0.80 MEN1 (0.68) MEN1KMT2AS100A4ESR1ESR2
SCHEMBL148272 0.80 ESR1 (0.42) ESR1ESR2NPC1
SCHEMBL6708180 0.79 MEN1 (0.56) MEN1KMT2AS100A4CYP3A4NFKB1
SCHEMBL726842 0.79 KDM4E (0.59) MEN1KMT2AESR1ALDH1A1POLB
SCHEMBL9358156 0.79 ALDH1A1 (0.64) MEN1KMT2AESR1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1660556-A1 COPOLYETHERIMIDES GENERAL ELECTRIC COMPANY (US) 2006-05-31 EP claimed
EP-1660560-A2 PHASE TRANSFER CATALYZED METHOD FOR PREPARATION OF POLYETEHRIMIDES GENERAL ELECTRIC COMPANY (US) 2006-05-31 EP claimed
WO-2005023901-A1 COPOLYETHERIMIDES GENERAL ELECTRIC COMPANY (US) 2005-03-17 WO claimed
WO-2005021618-A2 PHASE TRANSFER CATALYZED METHOD FOR PREPARATION OF POLYETEHRIMIDES GENERAL ELECTRIC COMPANY (US) 2005-03-10 WO claimed
US-6849706-B1 Copolyetherimides GENERAL ELECTRIC COMPANY (US) 2005-02-01 US claimed
EP-1660556-B1 COPOLYETHERIMIDES SABIC INNOVATIVE PLASTICS IP (NL) 2009-05-13 EP disclosed
EP-1403303-B1 Methods for the preparation of poly(etherimide)s GEN ELECTRIC (US) 2008-08-20 EP disclosed
EP-1660556-A1 COPOLYETHERIMIDES GENERAL ELECTRIC COMPANY (US) 2006-05-31 EP disclosed
EP-1426358-A3 Slurry preparation of bis(halophthalimides) and of polyether polymers GENERAL ELECTRIC COMPANY (US) 2006-03-08 EP disclosed
WO-2005023901-A1 COPOLYETHERIMIDES GENERAL ELECTRIC COMPANY (US) 2005-03-17 WO disclosed
US-6849706-B1 Copolyetherimides GENERAL ELECTRIC COMPANY (US) 2005-02-01 US disclosed
EP-1426358-A2 Slurry preparation of bis(halophthalimides) and of polyether polymers GENERAL ELECTRIC COMPANY (US) 2004-06-09 EP disclosed
EP-1222168-A2 SLURRY PREPARATION OF BIS(HALOPHTHALIMIDES) AND OF POLYETHER POLYMERS GENERAL ELECTRIC COMPANY (US) 2002-07-17 EP disclosed
WO-2001025196-A3 SLURRY PREPARATION OF BIS(HALOPHTHALIMIDES) AND OF POLYETHER POLYMERS GEN ELECTRIC (US) 2001-10-18 WO disclosed
US-6235866-B1 REACTING A DIAMINE, A HALOPHTHALIC ANHYDRIDE, AN ORGANIC LIQUID HAVING A POLARITY NO HIGHER THAN THAT OF O-DICHLOROBENZENE, DICHLOROTOLUENE, 1,2,4-TRICHLOROBENZENE, DIPHENYL SULFONE AND ANISOLE; AND AN IMIDIZATION CATALYST GENERAL ELECTRIC COMPANY 2001-05-22 US disclosed
WO-2001025196-A2 SLURRY PREPARATION OF BIS(HALOPHTHALIMIDES) AND OF POLYETHER POLYMERS GENERAL ELECTRIC COMPANY (US) 2001-04-12 WO disclosed