SCHEMBL3979000

SCHEMBL3979000

COc1cc(O)c(O)c(-n2nnc(OC(N)=O)c2-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
TMPRSS4 Q9NRS4 2/20 0.33
P2RX1 P51575 1/20 0.33
AKR1C3 P42330 1/20 0.33
RORB Q92753 1/20 0.33
KIF11 P52732 1/20 0.33
ADCY8 P40145 1/20 0.32
ADCY1 Q08828 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
XPO1 O14980 4/20 0.32
RECQL P46063 1/20 0.32
RUVBL1 Q9Y265 1/20 0.32
NPBWR1 P48145 1/20 0.31
MCHR1 Q99705 1/20 0.31
RBP4 P02753 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1344632 0.83 ALDH1A1 (0.36) ALDH1A1GAAAKR1C3RORBKIF11
SCHEMBL1148713 0.70 POLB (0.43) ALDH1A1GAAHSP90AA1XPO1
SCHEMBL679095 0.58 ALDH1A1 (0.50) ALDH1A1RXRARXRBRXRGTMPRSS4
SCHEMBL628410 0.58 PARP1 (0.50) GAARXRARXRBRXRGTMPRSS4
SCHEMBL31144953 0.58 PARP1 (0.50) GAARXRARXRBRXRGTMPRSS4
SCHEMBL5788396 0.58 RXRA (0.45) ALDH1A1RXRARXRBRXRGTMPRSS4
SCHEMBL29890062 0.58 RXRA (0.45) ALDH1A1RXRARXRBRXRGTMPRSS4
SCHEMBL28604363 0.57 KMT2A (0.50) ALDH1A1CYP3A4
SCHEMBL4762590 0.56 RXRA (0.48) ALDH1A1RXRARXRBRXRGTMPRSS4
SCHEMBL1147802 0.56 ABL1 (0.41) GAAHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054059-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-05-06 EP claimed
WO-2008021364-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2008-02-21 WO claimed