SCHEMBL3983370

SCHEMBL3983370

O=C(O)c1c(NS(=O)(=O)Cc2ccccc2)ccc2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 2/20 0.64
METAP1 P53582 1/20 0.64
ACLY P53396 1/20 0.50
HPGD P15428 4/20 0.49
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 3/20 0.49
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
HSD17B10 Q99714 2/20 0.49
GAA P10253 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
GLO1 Q04760 1/20 0.48
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
MMP1 P03956 1/20 0.45
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
MMP8 P22894 1/20 0.45
MMP13 P45452 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3979939 0.86 METAP2 (0.68) METAP2METAP1HPGDKDM4EALDH1A1
SCHEMBL3981564 0.82 METAP2 (0.63) METAP2METAP1HPGDKDM4EALDH1A1
SCHEMBL3985088 0.80 METAP2 (0.60) METAP2METAP1HPGDKDM4EALDH1A1
SCHEMBL3979514 0.80 METAP2 (0.60) METAP2METAP1PARP14
SCHEMBL3982567 0.80 METAP2 (0.71) METAP2METAP1HPGDKDM4EALDH1A1
SCHEMBL28028822 0.79 GLO1 (0.62) ACLYHPGDKDM4EALDH1A1KMT2A
SCHEMBL3986500 0.78 METAP2 (1.00) METAP2METAP1ALDH1A1KMT2AMEN1
SCHEMBL3985999 0.76 METAP2 (0.74) METAP2METAP1ACLYALDH1A1KMT2A
SCHEMBL7797715 0.75 ACLY (0.50) ACLYHPGDKDM4EALDH1A1KMT2A
SCHEMBL3978517 0.74 METAP2 (0.67) METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040068012-A1 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES 2004-04-08 US claimed
US-7491718-B2 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES (US) 2009-02-17 US disclosed
US-20040167128-A1 Sulfonamides having antiangiogenic and anticancer activity ABBVIE INC. 2004-08-26 US disclosed
US-20040157836-A1 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES 2004-08-12 US disclosed
US-20040068012-A1 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES 2004-04-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040167128-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP METAP2 1/4885METAP1 2/4885ACLY 2986/4885
US-20040068012-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP METAP2 1/4885METAP1 2/4885ACLY 2986/4885
US-20040157836-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP METAP2 1/4885METAP1 2/4885ACLY 2986/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.