SCHEMBL3985897

SCHEMBL3985897

Cc1c(Br)ccc(NS(=O)(=O)c2cccnc2)c1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 8/20 0.47
SLC40A1 Q9NP59 5/20 0.46
CKS1B P61024 3/20 0.46
SKP2 Q13309 3/20 0.46
GLO1 Q04760 1/20 0.45
METAP1 P53582 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
HTT P42858 1/20 0.44
BRD4 O60885 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3981261 0.86 ALDH1A1 (0.58) METAP2SLC40A1METAP1ALDH1A1GAA
SCHEMBL3979712 0.83 TP53 (0.47) CKS1BSKP2ALDH1A1
SCHEMBL3985688 0.83 CYP3A4 (0.49) METAP2SLC40A1CKS1BSKP2GLO1
SCHEMBL3983177 0.80 METAP2 (0.67) METAP2SLC40A1CKS1BSKP2GLO1
SCHEMBL3981344 0.79 METAP2 (0.56) METAP2METAP1ALDH1A1GAAHTT
SCHEMBL3985468 0.78 METAP2 (0.76) METAP2
SCHEMBL3984405 0.77 METAP2 (0.73) METAP2SLC40A1CKS1BSKP2GLO1
SCHEMBL25140692 0.73 ACLY (0.52) METAP2SLC40A1GLO1
SCHEMBL30806174 0.73 ACLY (0.52) METAP2SLC40A1GLO1
SCHEMBL16496135 0.73 ACLY (0.58) METAP2SLC40A1CKS1BSKP2GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7491718-B2 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES (US) 2009-02-17 US disclosed
EP-1549613-A1 SULFONAMIDES HAVING ANTIANGIOGENIC AND ANTICANCER ACTIVITY Abbott Laboratories (US) 2005-07-06 EP disclosed
US-20040167128-A1 Sulfonamides having antiangiogenic and anticancer activity ABBVIE INC. 2004-08-26 US disclosed
US-20040157836-A1 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES 2004-08-12 US disclosed
WO-2004033419-A1 SULFONAMIDES HAVING ANTIANGIOGENIC AND ANTICANCER ACTIVITY ABBOTT LABORATORIES (US) 2004-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040167128-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP METAP2 1/4885SLC40A1 3138/4885CKS1B 2502/4885
US-20040157836-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP METAP2 1/4885SLC40A1 3138/4885CKS1B 2502/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.