SCHEMBL3986499

SCHEMBL3986499

CNC(C(=O)NC(Cc1ccc(O)c(C(C)(C)C)c1)c1nccs1)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPRB P23467 3/20 0.40
CCR3 P51677 1/20 0.36
ADRB3 P13945 1/20 0.36
HSPA5 P11021 5/20 0.36
HSPA9 P38646 3/20 0.36
HSPA2 P54652 2/20 0.36
MRE11 P49959 1/20 0.34
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
LMNA P02545 1/20 0.33
XBP1 P17861 1/20 0.33
HSPA8 P11142 1/20 0.33
CNR2 P34972 1/20 0.33
CTSA P10619 1/20 0.32
TP53 P04637 1/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ACACB O00763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3987138 0.88 PTPRB (0.49) PTPRBHSPA5HSPA9HSPA2HTT
SCHEMBL3993082 0.88 PTPRB (0.40) PTPRBCCR3ADRB3HSPA5HSPA9
SCHEMBL3995134 0.83 ALOX12 (0.39) PTPRBCCR3ADRB3MRE11ALOX15
SCHEMBL13796750 0.83 PTPRB (0.36) PTPRBCCR3ADRB3HSPA5HSPA9
SCHEMBL3988530 0.83 PTPRB (0.36) PTPRBCCR3ADRB3HSPA5HSPA9
SCHEMBL3995019 0.81 PTPRB (0.38) PTPRBCCR3ADRB3HSPA5MRE11
SCHEMBL3995096 0.80 PTPRB (0.40) PTPRBADRB3
SCHEMBL4657375 0.79 ACACB (0.38) ALOX15ALOX12LMNATP53HTT
SCHEMBL3988336 0.78 PTPRB (0.46) PTPRBCCR3ADRB3
SCHEMBL3987548 0.77 ERCC1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553969-B1 Substituted phenethylamine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-06-30 US disclosed
EP-1149843-A1 SUBSTITUTED PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-10-31 EP disclosed