SCHEMBL4657375

SCHEMBL4657375

CNC(C(=O)NC(C)Cc1ccc(O)c(C(C)(C)C)c1)C(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.38
ALOX15 P16050 4/20 0.37
ALOX12 P18054 3/20 0.37
ALDH1A1 P00352 3/20 0.37
HSD17B10 Q99714 3/20 0.37
HSP90AA1 P07900 3/20 0.37
HSP90AB1 P08238 3/20 0.37
OPRK1 P41145 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 2/20 0.37
ESR1 P03372 2/20 0.37
TP53 P04637 2/20 0.37
CYP3A4 P08684 2/20 0.37
HPGD P15428 2/20 0.37
MAPK1 P28482 2/20 0.37
RECQL P46063 2/20 0.37
KMT2A Q03164 2/20 0.37
HIF1A Q16665 2/20 0.37
NR1I2 O75469 2/20 0.37
LMNA P02545 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3992083 0.81 NR1I2 (0.46) ALOX15ALDH1A1HSD17B10NR1I2LMNA
SCHEMBL4657426 0.80 KMT2A (0.38) ACACBALDH1A1OPRK1MEN1KMT2A
SCHEMBL4657437 0.80 KMT2A (0.38) ACACBALDH1A1OPRK1MEN1KMT2A
SCHEMBL3987561 0.79 MAPK1 (0.36) ACACBOPRK1MEN1MAPK1KMT2A
SCHEMBL3986499 0.79 PTPRB (0.40) ACACBALOX15ALOX12TP53LMNA
SCHEMBL3987548 0.79 ERCC1 (0.30) RENERCC1ERCC4
SCHEMBL3988356 0.79
SCHEMBL3989338 0.78 MMP1 (0.41) ALDH1A1MEN1KMT2ALMNARAB9A
SCHEMBL3988348 0.77 PTPRB (0.32) ALOX15ALOX12ALDH1A1HSD17B10HSP90AA1
SCHEMBL3988353 0.77 MMP13 (0.36) HSP90AA1HSP90AB1KDM4EMAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006122-B1 PHENETHYLAMINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2008-12-03 EP disclosed
US-6255285-B1 GASTROINTESTINAL DISORDERS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-07-03 US disclosed
EP-1006122-A1 PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-06-07 EP disclosed