SCHEMBL3987191

SCHEMBL3987191

CC(C)(C)c1ccc(OCC(=O)Nc2ccccc2C(=O)O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 1.00
MEN1 O00255 2/20 0.65
KMT2A Q03164 2/20 0.65
CASP3 P42574 1/20 0.65
SENP8 Q96LD8 1/20 0.65
SENP7 Q9BQF6 1/20 0.65
SENP6 Q9GZR1 1/20 0.65
TSHR P16473 2/20 0.62
MAPK10 P53779 2/20 0.62
ALDH1A1 P00352 2/20 0.62
HSD17B10 Q99714 1/20 0.62
POLB P06746 3/20 0.60
GAA P10253 1/20 0.60
CYP2C19 P33261 1/20 0.60
HIF1A Q16665 3/20 0.60
EPAS1 Q99814 2/20 0.60
RAB9A P51151 4/20 0.60
NPC1 O15118 3/20 0.60
KDM4E B2RXH2 1/20 0.58
SMN1; SMN2 Q16637 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6032429 0.86 HCAR2 (0.81) HCAR2MEN1KMT2ACASP3SENP8
SCHEMBL18510324 0.85 NPC1 (0.80) HCAR2MEN1KMT2ACASP3SENP8
SCHEMBL8689332 0.85 HCAR2 (1.00) HCAR2MEN1KMT2ACASP3SENP8
SCHEMBL8943790 0.85 HCAR2 (0.79) HCAR2MEN1KMT2ACASP3SENP8
SCHEMBL5696427 0.84 HCAR2 (0.78) HCAR2MEN1KMT2ACASP3SENP8
SCHEMBL5696407 0.83 HCAR2 (0.76) HCAR2MEN1KMT2ACASP3SENP8
SCHEMBL417809 0.83 HCAR2 (0.71) HCAR2MEN1KMT2AALDH1A1HSD17B10
SCHEMBL4914608 0.83 HCAR2 (0.76) HCAR2MEN1KMT2ACASP3SENP8
SCHEMBL4915695 0.83 HCAR2 (0.76) HCAR2MEN1KMT2ACASP3SENP8
SCHEMBL4912964 0.83 NPC1 (0.80) HCAR2MEN1KMT2ACASP3SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011057110-A1 GPR109A AGONISTS FOR THE TREATMENT OF CEREBRAL ISCHEMIA RUPRECHT-KARLS-UNIVERSITAT-HEIDELBERG (DE) 2011-05-12 WO disclosed
EP-2062578-A1 Novel use of chemical compounds for the treatment of AIDS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2009-05-27 EP disclosed
WO-2009063412-A1 USE OF CHEMICAL COMPOUNDS FOR THE TREATMENT OF AIDS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2009-05-22 WO disclosed